Oprelvekin

Table of contents

  • Brand Names
  • Chemistry
  • Pharmacologic Category
  • Mechanism of Action
  • Therapeutic Use
  • Pregnancy and Lactation Implications
  • Contraindications
  • Warnings and Precautions
  • Adverse Reactions
  • Genes that may be involved
  • Dosage
  • Pharmacokinetics and Pharmacodynamics
  • Special Considerations

Brand Names

North America

USA: Neumega.

Drug combinations

Chemistry

Oprelvekin: C~854~H~1411~N~253~O~235~S~2~. Mw: 19047.04. (1) 2-178-Interleukin 11 (human clone pXM/IL-11); (2) 2-178-Interleukin 11 (human clone pXM/IL-11). CAS-145941-26-0 (1996).

Pharmacologic Category

Hematopoietic Agents. Biological Response Modulator. Human Growth Factor. (ATC-Code: L03AC02).

Mechanism of action

Oprelvekin binds to the interleukin 11 receptor which leads to a cascade of signal transduction events. IL-11 is a thrombopoietic growth factor that directly stimulates the proliferation of hematopoietic stem cells and megakaryocyte progenitor cells and induces megakaryocyte maturation resulting in increased platelet production.

Therapeutic use

Prevention of severe thrombocytopenia. Reduction of need for platelet transfusions following myelosuppressive chemotherapy.

Pregnancy and lactiation implications

Adverse fetal effects in animals. There are no adequate studies in pregnant women. Use during pregnancy only if potential benefits outweigh potential risk to fetus. Excretion in breast milk unknown (use not recommended in nursing women).

Unlabeled use

Contraindications

Hypersensitivity to oprelvekin or any component of the formulation.

Warnings and precautions

Allergic or hypersensitivity reactions, including anaphylaxis, reported. Arrhythmia, pulmonary edema, and cardiac arrest reported (caution if history of atrial arrhythmia; may cause serious fluid retention; use cautiously in conditions where expansion of plasma volume should be avoided). Dose-limiting papilledema, more frequently associated with use in children, occurred (use with caution in pre-existing papilledema or with tumors involving CNS; patients experiencing oprelvekin-related papilledema have higher risk for visual acuity changes). Use with caution in pre-existing pericardial effusions or ascites, in hepatic/renal impairment, in respiratory disease, and in history of stroke or thromboembolic problems. Not indicated following myeloablative chemotherapy (higher risk of toxicity). Closely monitor fluid and electrolytes in patients on chronic diuretic therapy (severe hypokalemia may contribute to sudden death). May produce decreases in hemoglobin concentration, serum concentration of albumin and other proteins (result of expansion of plasma volume).

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